ONO-4059 analog

CAS No. 1351635-67-0

ONO-4059 analog( ONO 4059 analog | ONO4059 analog )

Catalog No. M11421 CAS No. 1351635-67-0

A highly potent and selective Btk inhibitor with IC50 in the sub-nM range; analog of ONO-4059.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 49 Get Quote
5MG 80 Get Quote
10MG 132 Get Quote
25MG 264 Get Quote
50MG 438 Get Quote
100MG 626 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    ONO-4059 analog
  • Note
    Research use only, not for human use.
  • Brief Description
    A highly potent and selective Btk inhibitor with IC50 in the sub-nM range; analog of ONO-4059.
  • Description
    A highly potent and selective Btk inhibitor with IC50 in the sub-nM range; analog of ONO-4059.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ONO 4059 analog | ONO4059 analog
  • Pathway
    Tyrosine Kinase
  • Target
    BTK
  • Recptor
    BTK
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1351635-67-0
  • Formula Weight
    456.4965
  • Molecular Formula
    C25H24N6O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 29 mg/mL
  • SMILES
    C=CC(=O)N1CCCC(C1)N2C3=NC=NC(=C3N(C2=O)C4=CC=C(C=C4)OC5=CC=CC=C5)N
  • Chemical Name
    8H-Purin-8-one, 6-amino-7,9-dihydro-9-[(3S)-1-(1-oxo-2-propen-1-yl)-3-piperidinyl]-7-(4-phenoxyphenyl)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Yamamoto, et al. WO 2011152351 A1 20111208.
molnova catalog
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